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- W3029791041 endingPage "2865" @default.
- W3029791041 startingPage "2852" @default.
- W3029791041 abstract "Opioid signaling plays a central role in pain perception. As such, it remains the main target in the development of antinociceptive agents, despite serious side effects involved. In recent years, hopes for improved opioid painkillers are rising, together with our understanding of allosterism and biased signaling mechanisms. In this review, we focus on recently discovered allosteric modulators of opioid receptors, insights into phenomena underlying their action, as well as on how they extend our understanding of mechanisms of previously known compounds. A brief overlook of their synthesis is also presented." @default.
- W3029791041 created "2020-06-05" @default.
- W3029791041 creator A5025358484 @default.
- W3029791041 creator A5036909810 @default.
- W3029791041 creator A5059100019 @default.
- W3029791041 creator A5071363313 @default.
- W3029791041 date "2020-12-03" @default.
- W3029791041 modified "2023-10-02" @default.
- W3029791041 title "Tuning Down the Pain – An Overview of Allosteric Modulation of Opioid Receptors: Mechanisms of Modulation, Allosteric Sites, Modulator Syntheses" @default.
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