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- W3030571330 endingPage "699" @default.
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- W3030571330 abstract "临床工作中发现,要使患者血中他克莫司(FK506)的浓度达到有效范围,个体间的FK506用量差异较大.据文献报道,这种区别在不同种族之间尤为明显,一般来说,黑人的用药剂量要高于其他种族2倍以上[1-3].这种区别主要是因FK506吸收差异而不是清除差异造成的,而吸收的障碍主要受药物代谢酶P450(CYP)以及多重耐药基因MDR1所编码的P糖蛋白的影响.FK506在体内主要是由P450亚家族(主要包括CYP3A4和CYP3A5)代谢。" @default.
- W3030571330 created "2020-06-05" @default.
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- W3030571330 date "2005-11-20" @default.
- W3030571330 modified "2023-09-25" @default.
- W3030571330 title "肾移植患者血他克莫司浓度/剂量比与CYP 3A5基因多态性的关系" @default.
- W3030571330 doi "https://doi.org/10.3760/cma.j.issn.0254-1785.2005.11.020" @default.
- W3030571330 hasPublicationYear "2005" @default.
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