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- W3036700967 endingPage "105018" @default.
- W3036700967 startingPage "105018" @default.
- W3036700967 abstract "Stroke is a major cause of mortality and morbidity worldwide. Considerable experimental and clinical evidence suggests that both diabetes mellitus (DM) and post-stroke hyperglycemia are associated with increased mortality rate and worsened clinical conditions in acute ischemic stroke (AIS) patients. Insulin treatment does not seem to provide convincing benefits for these patients, therefore prompting a change of strategy. The selective agonists of Glucagon-Like Peptide-1 Receptors (GLP-1Ras) and the Inhibitors of Dipeptidyl Peptidase-IV (DPP-IVIs, gliptins) are two newer classes of glucose-lowering drugs used for the treatment of DM. This review examines in detail the rationale for their development and the physicochemical, pharmacokinetic and pharmacodynamic properties and clinical activities. Emphasis will be placed on their neuroprotective effects at cellular and molecular levels in experimental models of acute cerebral ischemia. In perspective, an adequate basis does exist for a novel therapeutic approach to hyperglycemia in AIS patients through the additive treatment with GLP-1Ras plus DPP-IVIs." @default.
- W3036700967 created "2020-06-25" @default.
- W3036700967 creator A5024268953 @default.
- W3036700967 creator A5052622611 @default.
- W3036700967 creator A5059939846 @default.
- W3036700967 date "2020-10-01" @default.
- W3036700967 modified "2023-10-17" @default.
- W3036700967 title "The treament of hyperglycemia in acute ischemic stroke with incretin-based drugs" @default.
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