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- W3040888857 endingPage "1753" @default.
- W3040888857 startingPage "1744" @default.
- W3040888857 abstract "In contrast to other drug-metabolizing cytochrome P450 (CYP) oxygenases, CYP2J2 shows considerable extrahepatic activity and is responsible for the olefin epoxidation of several polyunsaturated fatty acid (PUFA) precursors. The resulting epoxylipids act as signaling mediators and show a remarkable variety of biological functions. Recent studies suggest a role of selected CYP2J2-derived epoxylipids and their metabolites in chronic pain, as well as angiogenesis, hematopoiesis, metabolic disorders, and tumor growth. These pleiotropic effects of CYP products imply that targeting CYP2J2 could represent a novel therapeutic strategy in these fields. Here, we explore the biological functions of CYP2J2-derived epoxylipids and discuss therapeutic implications of the CYP2J2 inhibitors that are known so far." @default.
- W3040888857 created "2020-07-16" @default.
- W3040888857 creator A5017526919 @default.
- W3040888857 creator A5066815637 @default.
- W3040888857 creator A5078612562 @default.
- W3040888857 creator A5082078699 @default.
- W3040888857 date "2020-09-01" @default.
- W3040888857 modified "2023-09-27" @default.
- W3040888857 title "Exploring CYP2J2: lipid mediators, inhibitors and therapeutic implications" @default.
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- W3040888857 doi "https://doi.org/10.1016/j.drudis.2020.07.002" @default.
- W3040888857 hasPubMedId "https://pubmed.ncbi.nlm.nih.gov/32652311" @default.
- W3040888857 hasPublicationYear "2020" @default.
- W3040888857 type Work @default.