Matches in SemOpenAlex for { <https://semopenalex.org/work/W3042934810> ?p ?o ?g. }
- W3042934810 endingPage "2103" @default.
- W3042934810 startingPage "2090" @default.
- W3042934810 abstract "Dysregulated inflammation is a central pathological process in diverse disease states, including neurodegenerative disorders. The recent concept of “resolution of inflammation” is offering a conceptual change for the diagnosis and the development of new therapeutic approaches for chronic inflammatory diseases. Resolution of inflammation terminates the inflammatory response promoting the return to tissue homeostasis through the action of several classes of mediators, termed specialized pro-resolving lipid mediators (SPMs), that include lipoxins, resolvins, protectins, and maresins. SPMs provide “stop signals” that reduce the number of immune cells at the site of insult and increase the clearance of apoptotic cells through phagocytosis. SPMs elicit their effects through the interaction with specific G-protein coupled receptors (GPCRs). The elucidation of the pathways downstream of the GPCRs involved in the resolution of chronic inflammation is opening novel opportunities to generate novel anti-inflammatory agents. This review focuses on the SPMs and the receptors through which their effects are mediated. The medicinal chemistry of the modulators of the GPCRs involved in the resolution of inflammation will be illustrated, by highlighting the potential for developing new antiinflammatory drugs." @default.
- W3042934810 created "2020-07-23" @default.
- W3042934810 creator A5010068826 @default.
- W3042934810 creator A5021058541 @default.
- W3042934810 creator A5029727582 @default.
- W3042934810 creator A5082844616 @default.
- W3042934810 date "2021-01-14" @default.
- W3042934810 modified "2023-09-23" @default.
- W3042934810 title "G-Protein Coupled Receptors Involved in the Resolution of Inflammation: Ligands and Therapeutic Perspectives" @default.
- W3042934810 cites W1194718656 @default.
- W3042934810 cites W1497700962 @default.
- W3042934810 cites W1544184390 @default.
- W3042934810 cites W1554897154 @default.
- W3042934810 cites W1964051296 @default.
- W3042934810 cites W1964054981 @default.
- W3042934810 cites W1974309015 @default.
- W3042934810 cites W1976768202 @default.
- W3042934810 cites W1981748455 @default.
- W3042934810 cites W1983795363 @default.
- W3042934810 cites W1984554579 @default.
- W3042934810 cites W1986483382 @default.
- W3042934810 cites W1988697119 @default.
- W3042934810 cites W1990014836 @default.
- W3042934810 cites W1991047945 @default.
- W3042934810 cites W1991494867 @default.
- W3042934810 cites W1999224453 @default.
- W3042934810 cites W2003741314 @default.
- W3042934810 cites W2007749067 @default.
- W3042934810 cites W2010972120 @default.
- W3042934810 cites W2011885150 @default.
- W3042934810 cites W2014462125 @default.
- W3042934810 cites W2026708741 @default.
- W3042934810 cites W2030691041 @default.
- W3042934810 cites W2035641637 @default.
- W3042934810 cites W2036359942 @default.
- W3042934810 cites W2039694091 @default.
- W3042934810 cites W2044609482 @default.
- W3042934810 cites W2052852012 @default.
- W3042934810 cites W2073926013 @default.
- W3042934810 cites W2083041617 @default.
- W3042934810 cites W2084117223 @default.
- W3042934810 cites W2090609282 @default.
- W3042934810 cites W2090956219 @default.
- W3042934810 cites W2098965240 @default.
- W3042934810 cites W2100607138 @default.
- W3042934810 cites W2101291779 @default.
- W3042934810 cites W2103010344 @default.
- W3042934810 cites W2103448780 @default.
- W3042934810 cites W2107104127 @default.
- W3042934810 cites W2108943513 @default.
- W3042934810 cites W2109326384 @default.
- W3042934810 cites W2119001835 @default.
- W3042934810 cites W2120699390 @default.
- W3042934810 cites W2122523355 @default.
- W3042934810 cites W2123991105 @default.
- W3042934810 cites W2128829928 @default.
- W3042934810 cites W2131896212 @default.
- W3042934810 cites W2140210316 @default.
- W3042934810 cites W2140526459 @default.
- W3042934810 cites W2145164843 @default.
- W3042934810 cites W2148536296 @default.
- W3042934810 cites W2152145035 @default.
- W3042934810 cites W2161273513 @default.
- W3042934810 cites W2163134721 @default.
- W3042934810 cites W2166487622 @default.
- W3042934810 cites W2168256748 @default.
- W3042934810 cites W2168879708 @default.
- W3042934810 cites W2171245653 @default.
- W3042934810 cites W2206288859 @default.
- W3042934810 cites W2210741139 @default.
- W3042934810 cites W2295384369 @default.
- W3042934810 cites W2298859064 @default.
- W3042934810 cites W2333427125 @default.
- W3042934810 cites W2339222516 @default.
- W3042934810 cites W2416672343 @default.
- W3042934810 cites W2472659787 @default.
- W3042934810 cites W2507972426 @default.
- W3042934810 cites W2517461385 @default.
- W3042934810 cites W2520447320 @default.
- W3042934810 cites W2535933709 @default.
- W3042934810 cites W2565125046 @default.
- W3042934810 cites W2587567454 @default.
- W3042934810 cites W2597925028 @default.
- W3042934810 cites W2752260686 @default.
- W3042934810 cites W2755916089 @default.
- W3042934810 cites W2766158825 @default.
- W3042934810 cites W2785252094 @default.
- W3042934810 cites W2791354060 @default.
- W3042934810 cites W2801066468 @default.
- W3042934810 cites W2805396917 @default.
- W3042934810 cites W2892306013 @default.
- W3042934810 cites W2897027772 @default.
- W3042934810 cites W2898668843 @default.
- W3042934810 cites W2900408032 @default.
- W3042934810 cites W2901773763 @default.
- W3042934810 cites W2904995365 @default.
- W3042934810 cites W2943831945 @default.
- W3042934810 cites W2970729530 @default.