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- W3094671567 endingPage "17" @default.
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- W3094671567 abstract "A large number of cannabinoids have been discovered that could play a role in mitigating cardiac affections. However, none of them has been as widely studied as cannabidiol (CBD), most likely because, individually, the others offer only partial effects or can activate potential harmful pathways. In this regard, CBD has proven to be of great value as a cardioprotective agent since it is a potent antioxidant and anti-inflammatory molecule. Thus, we conducted a review to condensate the currently available knowledge on CBD as a therapy for different experimental models of cardiomyopathies and heart failure to detect the molecular pathways involved in cardiac protection. CBD therapy can greatly limit the production of oxygen/nitrogen reactive species, thereby limiting cellular damage, protecting mitochondria, avoiding caspase activation, and regulating ionic homeostasis. Hence, it can affect myocardial contraction by restricting the activation of inflammatory pathways and cytokine secretion, lowering tissular infiltration by immune cells, and reducing the area of infarct and fibrosis formation. These effects are mediated by the activation or inhibition of different receptors and target molecules of the endocannabinoid system. In the final part of this review, we explore the current state of CBD in clinical trials as a treatment for cardiovascular diseases and provide evidence of its potential benefits in humans." @default.
- W3094671567 created "2020-11-09" @default.
- W3094671567 creator A5016153880 @default.
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- W3094671567 creator A5045279875 @default.
- W3094671567 creator A5069071467 @default.
- W3094671567 creator A5084721186 @default.
- W3094671567 date "2020-10-27" @default.
- W3094671567 modified "2023-10-15" @default.
- W3094671567 title "Therapeutic Applications of Cannabinoids in Cardiomyopathy and Heart Failure" @default.
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