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- W3113118133 abstract "This chapter describes the research program that led to the discovery of vixotrigine, a use-dependent voltage-gated sodium channel blocker designed to deliver an improved safety profile. The properties that led to the selection of this candidate molecule are discussed. The choice of initial synthetic strategy and the development of an early scalable synthesis are examined. Further development of a more efficient process and the incorporation of green chemistry principles to successfully prepare for commercial utility are described." @default.
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- W3113118133 date "2020-01-01" @default.
- W3113118133 modified "2023-10-13" @default.
- W3113118133 title "Discovery and Chemical Development of the Use-Dependent Sodium Channel Blocker Vixotrigine for the Treatment of Pain" @default.
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