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- W3119780493 abstract "Biologic medicines are designed rationally based on an understanding of the complex biochemical and physiologic pathways in a disease state. Understanding the structure and function of key protein molecules in these pathways (drug targets) has transformed the discovery and development paradigm of biologic medicines. In this chapter, the biochemical, physiologic, and pharmacological basis of biologic medicines are discussed, based on the most common major targets of biologics as adopted during the drug discovery process. The human epidermal growth factor family (HER) is a group of receptor tyrosine kinases (RTKs) that comprise four members: HER1, HER2, HER3, and HER4. The human vascular endothelial growth factor (VEGF) family comprises of five members, VEGF-A (commonly known as VEGF), VEGF-B, VEGF-C, VEGF-D, and placental growth factor (PlGF); VEGF is the most studied and clinically relevant. Interleukins consist of more than 60 potent pro-inflammatory pleiotropic (having multiple effects) cytokines." @default.
- W3119780493 created "2021-01-18" @default.
- W3119780493 creator A5004913828 @default.
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- W3119780493 creator A5067632543 @default.
- W3119780493 creator A5088845547 @default.
- W3119780493 date "2020-12-30" @default.
- W3119780493 modified "2023-10-18" @default.
- W3119780493 title "Drug Targets for Biologics" @default.
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