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- W3124183720 endingPage "67" @default.
- W3124183720 startingPage "67" @default.
- W3124183720 abstract "Antifungal drugs and antifungal agrochemicals have significant limitations. These include several unintended consequences of their use including the growing importance of intrinsic and acquired resistance. These problems underpin an increasingly urgent need to improve the existing classes of antifungals and to discover novel antifungals. Structural insights into drug targets and their complexes with both substrates and inhibitory ligands increase opportunity for the discovery of more effective antifungals. Implementation of this promise, which requires multiple skill sets, is beginning to yield candidates from discovery programs that could more quickly find their place in the clinic. This review will describe how structural biology is providing information for the improvement and discovery of inhibitors targeting the essential fungal enzyme sterol 14α-demethylase." @default.
- W3124183720 created "2021-02-01" @default.
- W3124183720 creator A5010888782 @default.
- W3124183720 creator A5055005364 @default.
- W3124183720 date "2021-01-20" @default.
- W3124183720 modified "2023-09-26" @default.
- W3124183720 title "Roles for Structural Biology in the Discovery of Drugs and Agrochemicals Targeting Sterol 14α-Demethylases" @default.
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