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- W3133670261 endingPage "597" @default.
- W3133670261 startingPage "597" @default.
- W3133670261 abstract "Since the seminal breakthrough of treating diabetic patients with insulin in the 1920s, there has been great interest in developing other proteins and their peptide mimetics as therapies for a wide variety of other medical disorders. Currently, there are at least 60 different peptides that have been approved for human use and over 150 peptides that are in various stages of clinical development. Peptides mimetic of the major proteins on lipoproteins, namely apolipoproteins, have also been developed first as tools for understanding apolipoprotein structure and more recently as potential therapeutics. In this review, we discuss the biochemistry, peptide mimetics design and clinical trials for peptides based on apoA-I, apoE and apoC-II. We primarily focus on applications of peptide mimetics related to cardiovascular diseases. We conclude with a discussion on the limitations of peptides as therapeutic agents and the challenges that need to be overcome before apolipoprotein mimetic peptides can be developed into new drugs." @default.
- W3133670261 created "2021-03-15" @default.
- W3133670261 creator A5011350352 @default.
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- W3133670261 creator A5040295868 @default.
- W3133670261 creator A5045047702 @default.
- W3133670261 creator A5068951391 @default.
- W3133670261 date "2021-03-08" @default.
- W3133670261 modified "2023-10-02" @default.
- W3133670261 title "Apolipoprotein Mimetic Peptides: Potential New Therapies for Cardiovascular Diseases" @default.
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