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- W3136772521 startingPage "275" @default.
- W3136772521 abstract "Oxycodone is a semisynthetic μ- and κ-opioid receptor with agonist with a broad scope of use including postoperative analgesia as well as control of neuropathic and cancer pain. Advantages over other opioids include prolonged duration of action, greater potency than morphine and lack of histamine release or ceiling effect. Individual responses to oxycodone can vary due to genetic differences. This review article aims to summarize the oxycodone literature and provide context on its pharmacogenomics and pharmacokinetics. The evidence for clinical effect of genetic polymorphisms on oxycodone is conflicting. There is stronger evidence linking polymorphic genetic enzymes CYP2D6 and CYP3A with therapeutic outcomes. Further, research is needed to discern all of oxycodone's metabolites and their contribution to the overall analgesic effect." @default.
- W3136772521 created "2021-03-29" @default.
- W3136772521 creator A5062638610 @default.
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- W3136772521 creator A5067360995 @default.
- W3136772521 creator A5074073608 @default.
- W3136772521 creator A5075340457 @default.
- W3136772521 date "2021-04-01" @default.
- W3136772521 modified "2023-10-14" @default.
- W3136772521 title "Pharmacogenomics of oxycodone: a narrative literature review" @default.
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