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• W3137229084 endingPage "1014" @default.
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• W3137229084 abstract "A practical and scalable route to (3aR, 9bR)-8-fluoro-7-(perfluoropropan-2-yl)-9b-(phenylsulfonyl)-2,3,3a,4,5,9b-hexahydro-1H-benzo[e]indole 10, an advanced intermediate en route to the synthesis of the RORγt inverse agonist, BMT-362265, is described starting from fluorobenzene. The synthesis involved the screening of multiple synthetic routes for their feasibility and scalability. We also demonstrate the utility of an annulating reagent, (R)-N-(2-chloroethyl)-2-methylpropane-2-sulfinamide, for the diastereoselective synthesis of tricyclic pyrrolidine intermediates 24 and 36 on a multigram scale." @default.
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• W3137229084 date "2021-03-16" @default.
• W3137229084 modified "2023-10-16" @default.
• W3137229084 title "Practical Synthesis of (3a<i>R</i>, 9b<i>R</i>)-8-Fluoro-7-(perfluoropropan-2-yl)-9b-(phenylsulfonyl)-2,3,3a,4,5,9b-hexahydro-1<i>H</i>-benzo[e]indole: An Advanced Intermediate to Access the RORγt Inverse Agonist <b>BMT-362265</b>" @default.
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• W3137229084 doi "https://doi.org/10.1021/acs.oprd.1c00019" @default.
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