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- W3137451702 endingPage "105572" @default.
- W3137451702 startingPage "105572" @default.
- W3137451702 abstract "Metabolic diseases are becoming increasingly common in modern society. Therefore, it is essential to develop effective drugs or new treatments for metabolic diseases. As an active ingredient derived from plants, celastrol has shown great potential in the treatment of a wide variety of metabolic diseases and received considerable attention in recent years. In reported studies, the anti-obesity effect of celastrol resulted from regulating leptin sensitivity, energy metabolism, inflammation, lipid metabolism and even gut microbiota. Celastrol reversed insulin resistance via multiple routes to protect against type 2 diabetes. Celastrol also showed effects on atherosclerosis, cholestasis and osteoporosis. Celastrol in treating metabolic diseases seem to be versatile and the targets or pathways were diverse. Here, we systematically review the mechanism of action, and the therapeutic properties of celastrol in various metabolic diseases and complications. Based on this review, potential research strategies might contribute to the celastrol's clinical application in the future." @default.
- W3137451702 created "2021-03-29" @default.
- W3137451702 creator A5002603423 @default.
- W3137451702 creator A5009247381 @default.
- W3137451702 creator A5015956915 @default.
- W3137451702 creator A5033954071 @default.
- W3137451702 creator A5077518155 @default.
- W3137451702 creator A5081787708 @default.
- W3137451702 creator A5088357346 @default.
- W3137451702 date "2021-05-01" @default.
- W3137451702 modified "2023-10-14" @default.
- W3137451702 title "Celastrol in metabolic diseases: Progress and application prospects" @default.
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