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- W3137792315 abstract "Simultaneous inhibition of tumors and tumor metastasis can be considered as an ideal and ultimate goal for cancer therapy. We report a unique platform based on DNA aptamer-functionalized microfibrous rings for simultaneous inhibition of primary tumors and tumor metastasis. Doxorubicin-loaded electrospun poly(lactic-co-glycolic acid) fibrous mat was prepared and homogenized in the presence of salt to form microfibrous rings that were functionalized with gadolinium chelates and DNA aptamer via polyethyleneimine-mediated conjugation. The multifunctional fibrous rings have an average diameter of 11.1 µm, and exhibit good biocompatibility, pH-dependent long-term drug release profile, and a high r1 relaxivity. Due to the ring structure and the DNA aptamer functionalization, the multifunctional fibrous rings are able to target and anchor tumor cells for a relatively long retention time as verified by magnetic resonance imaging, consequently decreasing the tumor cell shedding into the blood to form circulating tumor cells and inhibiting tumor metastasis and invasion." @default.
- W3137792315 created "2021-03-29" @default.
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- W3137792315 date "2021-06-01" @default.
- W3137792315 modified "2023-09-30" @default.
- W3137792315 title "Multifunctional PLGA microfibrous rings enable MR imaging-guided tumor chemotherapy and metastasis inhibition through prevention of circulating tumor cell shedding" @default.
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- W3137792315 doi "https://doi.org/10.1016/j.nantod.2021.101123" @default.
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