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- W3140149191 abstract ") 价值分别地是 26, 20,和 18 μmol/L。为 24 h 的 10, 20,和 40 μmol/L ursolic 酸治疗的 apoptotic 率是 5.74% , 14.49% ,和 33.05% ,并且为 48, h 分别地是 9% , 21.39% ,和 40.49% 。Ursolic 酸压制了 EGFR, ERK1/2, p38 MAPK,和 JNK 的 phosphorylation,它很好与它的生长被相关禁止的效果。10, 20,和 40 μmol/L ursolic 酸显著地禁止了刺激 EGF 的 HT-29 房间(P<0.05 ) 的增长。当与酸与 200 nmol/L AG 1478 或 10 μmol/L U0126 (P<0.01 ) 相结合的 10 和 20 μmol/L ursolic 对待时,房间增长最显著地被禁止。而且,它也下面调整 Bcl-2 和 Bcl-xL 和激活的 caspase-3 和 caspase-9 的表示。结论 Ursolic 酸由压制 EGFR/MAPK 小径在 HT-29 房间导致 apoptosis,建议它可以是为颜色的治疗的一个有势力代理人表面的癌症。" @default.
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- W3140149191 date "2009-01-01" @default.
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- W3140149191 title "Ursolic acid inhibits proliferation and induces apoptosis of HT-29 colon cancer cells by inhibiting the EGFR/MAPK pathway" @default.
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