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- W3146845599 abstract "Motivation. Complexes between nucleic acids and phospholipid vesicles have been developed as stable non– viral gene delivery vehicles. Currently employed approach uses positively charged lipid species and a helper zwitterionic lipid, the latter being applied for the stabilization of the whole complex. However, besides problematic steps during their preparation, cationic lipids are toxic for cells. The present work describes some energetic issues pertinent to preparation and use of neutral lipid–DNA self–assemblies, thus avoiding toxicity of lipoplexes. Thermodynamic measurements showed stabilization of polynucleotide helix upon its interaction with liposomes in the presence of divalent metal cations. It is thus possible to suggest this self–assembly as an improved formulation for use in gene delivery. Method. Thermotropic phase transitions of zwitterionic liposomes and their complexes with DNA in the presence of Mg 2+" @default.
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- W3146845599 date "2004-01-01" @default.
- W3146845599 modified "2023-09-27" @default.
- W3146845599 title "Divalent Cation Induced DNA-Zwitterionic Vesicle Formulation Compacted for Gene Delivery: Thermodynamic Aspects #" @default.
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