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- W3148865513 abstract "简化 aminocoumarin 类似物,任何一个 noviosylated 或简单基本 heterocycle 依附 3-amido-coumarin 混合物,被知道正在答应 anticancer 代理人指向 Hsp90 的 C 终端 ATP 有约束力的地点。在这研究,在包含 Hsp90 C 终端禁止者的二已知的 noviose 的 noviose 一半的 3-amino isosteric 代替综合地第一次被认识到。在这些的 vitro 评估,混合物建议进 noviose 子单元的一个基本的氨基的组的介绍导致了他们的 cytotoxicities 的重要改进。" @default.
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- W3148865513 date "2013-01-01" @default.
- W3148865513 modified "2023-10-13" @default.
- W3148865513 title "Simplified aminocoumarin analogues as anticancer agents:Amino isosteric replacement in the noviose moiety resulted in substantial enhancement of antiproliferative activity" @default.
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