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- W3150422034 endingPage "95" @default.
- W3150422034 startingPage "63" @default.
- W3150422034 abstract "Epigenetic writers, erasers, and readers are the targets of drugs that are FDA-approved or in clinical trials. Classical chemical strategies have been employed to discover these new chemical agents. We illustrate herein through several examples the rational drug design approaches, the screening assays, and the chemical optimization that led to their discovery. Finally, we describe the pharmacological assays that were set-up for the preclinical profiling of epigenetic drugs and provide open questions on how difficult it is to target epigenetic enzymes and readers in drug development." @default.
- W3150422034 created "2021-04-13" @default.
- W3150422034 creator A5008017948 @default.
- W3150422034 creator A5031452617 @default.
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- W3150422034 creator A5045822769 @default.
- W3150422034 creator A5054568991 @default.
- W3150422034 creator A5078177483 @default.
- W3150422034 date "2016-01-01" @default.
- W3150422034 modified "2023-10-16" @default.
- W3150422034 title "Drug Discovery Methods" @default.
- W3150422034 cites W1027568982 @default.
- W3150422034 cites W1963736125 @default.
- W3150422034 cites W1964746150 @default.
- W3150422034 cites W1964767882 @default.
- W3150422034 cites W1966164805 @default.
- W3150422034 cites W1966590731 @default.
- W3150422034 cites W1967764418 @default.
- W3150422034 cites W1969807932 @default.
- W3150422034 cites W1970517458 @default.
- W3150422034 cites W1970675267 @default.
- W3150422034 cites W1971004265 @default.
- W3150422034 cites W1971273543 @default.
- W3150422034 cites W1972635017 @default.
- W3150422034 cites W1977199336 @default.
- W3150422034 cites W1978319260 @default.
- W3150422034 cites W1978660434 @default.
- W3150422034 cites W1979142801 @default.
- W3150422034 cites W1980937575 @default.
- W3150422034 cites W1981259130 @default.
- W3150422034 cites W1982619775 @default.
- W3150422034 cites W1986042567 @default.
- W3150422034 cites W1988594891 @default.
- W3150422034 cites W1989186239 @default.
- W3150422034 cites W1990931780 @default.
- W3150422034 cites W1992288855 @default.
- W3150422034 cites W1995204800 @default.
- W3150422034 cites W1995275377 @default.
- W3150422034 cites W1995557117 @default.
- W3150422034 cites W1995827055 @default.
- W3150422034 cites W1995895091 @default.
- W3150422034 cites W1997275786 @default.
- W3150422034 cites W1998351475 @default.
- W3150422034 cites W2000156285 @default.
- W3150422034 cites W2004380688 @default.
- W3150422034 cites W2005829971 @default.
- W3150422034 cites W2006500779 @default.
- W3150422034 cites W2010899127 @default.
- W3150422034 cites W2011104528 @default.
- W3150422034 cites W2011453131 @default.
- W3150422034 cites W2013154874 @default.
- W3150422034 cites W2013810007 @default.
- W3150422034 cites W2014107899 @default.
- W3150422034 cites W2015134259 @default.
- W3150422034 cites W2015215119 @default.
- W3150422034 cites W2015475080 @default.
- W3150422034 cites W2017492512 @default.
- W3150422034 cites W2018366426 @default.
- W3150422034 cites W2024373518 @default.
- W3150422034 cites W2024713471 @default.
- W3150422034 cites W2025006523 @default.
- W3150422034 cites W2029124536 @default.
- W3150422034 cites W2031441006 @default.
- W3150422034 cites W2031810803 @default.
- W3150422034 cites W2032191311 @default.
- W3150422034 cites W2032365395 @default.
- W3150422034 cites W2032743020 @default.
- W3150422034 cites W2033102369 @default.
- W3150422034 cites W2038564831 @default.
- W3150422034 cites W2040074276 @default.
- W3150422034 cites W2040092511 @default.
- W3150422034 cites W2040263155 @default.
- W3150422034 cites W2040393829 @default.
- W3150422034 cites W2041535798 @default.
- W3150422034 cites W2046588282 @default.
- W3150422034 cites W2048389974 @default.
- W3150422034 cites W2048617427 @default.
- W3150422034 cites W2051469259 @default.
- W3150422034 cites W2053213384 @default.
- W3150422034 cites W2054301876 @default.
- W3150422034 cites W2054696920 @default.
- W3150422034 cites W2055276981 @default.
- W3150422034 cites W2055770867 @default.
- W3150422034 cites W2056842797 @default.
- W3150422034 cites W2057529572 @default.
- W3150422034 cites W2060424322 @default.
- W3150422034 cites W2060596553 @default.
- W3150422034 cites W2061819850 @default.
- W3150422034 cites W2062768506 @default.
- W3150422034 cites W2062828530 @default.
- W3150422034 cites W2063296278 @default.
- W3150422034 cites W2063887542 @default.
- W3150422034 cites W2065125513 @default.
- W3150422034 cites W2068739830 @default.
- W3150422034 cites W2073113196 @default.
- W3150422034 cites W2074287116 @default.
- W3150422034 cites W2078616374 @default.
- W3150422034 cites W2079392960 @default.