Matches in SemOpenAlex for { <https://semopenalex.org/work/W3164284040> ?p ?o ?g. }
- W3164284040 endingPage "149" @default.
- W3164284040 startingPage "133" @default.
- W3164284040 abstract "The internalization of G protein-coupled receptors (GPCRs) is an important mechanism regulating the signal strength and limiting the opportunity of receptor activation. Based on the importance of GPCRs, the detailed knowledge about the regulation of signal transduction is crucial. Here, current knowledge about the agonist-induced, arrestin-dependent internalization process of rhodopsin-like GPCRs is reviewed. Arrestins are conserved molecules that act as key players within the internalization process of many GPCRs. Based on highly conserved structural characteristics within the rhodopsin-like GPCRs, the identification of arrestin interaction sites in model systems can be compared and used for the investigation of internalization processes of other receptors. The increasing understanding of this essential regulation mechanism of receptors can be used for drug development targeting rhodopsin-like GPCRs. Here, we focus on the neuropeptide Y receptor family, as these receptors transmit various physiological processes such as food intake, energy homeostasis, and regulation of emotional behavior, and are further involved in pathophysiological processes like cancer, obesity and mood disorders. Hence, this receptor family represents an interesting target for the development of novel therapeutics requiring the understanding of the regulatory mechanisms influencing receptor mediated signaling." @default.
- W3164284040 created "2021-06-07" @default.
- W3164284040 creator A5056535488 @default.
- W3164284040 creator A5057051630 @default.
- W3164284040 creator A5073399193 @default.
- W3164284040 date "2021-05-26" @default.
- W3164284040 modified "2023-09-26" @default.
- W3164284040 title "Arrestin-dependent internalization of rhodopsin-like G protein-coupled receptors" @default.
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