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- W3185483707 endingPage "110092" @default.
- W3185483707 startingPage "110092" @default.
- W3185483707 abstract "Cell surface receptors including the epidermal growth factor receptor (EGFR) family and G-protein coupled receptors (GPCRs) play quintessential roles in physiology, and in diseases, including cardiovascular diseases. While downstream signaling from these individual receptor families has been well studied, the cross-talk between EGF and GPCR receptor families is still incompletely understood. Including members of both receptor families, the number of receptor and ligand combinations for unique interactions is vast, offering a frontier of pharmacologic targets to explore for preventing and treating disease. This molecular cross-talk, called receptor transactivation, is reviewed here with a focus on the cardiovascular system featuring the well-studied GPCR receptors, but also discussing less-studied receptors from both families for a broad understanding of context of expansile interactions, repertoire of cellular signaling, and disease consequences. Attention is given to cell type, level of chronicity, and disease context given that transactivation and comorbidities, including diabetes, hypertension, coronavirus infection, impact cardiovascular disease and health outcomes." @default.
- W3185483707 created "2021-08-02" @default.
- W3185483707 creator A5047153131 @default.
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- W3185483707 creator A5056281943 @default.
- W3185483707 creator A5060445649 @default.
- W3185483707 creator A5061040306 @default.
- W3185483707 date "2021-10-01" @default.
- W3185483707 modified "2023-10-16" @default.
- W3185483707 title "GPCR-ErbB transactivation pathways and clinical implications" @default.
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