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- W3186346120 abstract "N6-methyladenosine (m6A) has emerged as an abundant modification throughout the transcriptome with widespread functions in protein-coding and noncoding RNAs. It affects the fates of modified RNAs, including their stability, splicing, and/or translation, and thus plays important roles in posttranscriptional regulation. To date, m6A methyltransferases have been reported to execute m6A deposition on distinct RNAs by their own or forming different complexes with additional partner proteins. In this review, we summarize the function of these m6A methyltransferases or complexes in regulating the key genes and pathways of cancer biology. We also highlight the progress in the use of m6A methyltransferases in mediating therapy resistance, including chemotherapy, targeted therapy, immunotherapy and radiotherapy. Finally, we discuss the current approaches and clinical potential of m6A methyltransferase-targeting strategies." @default.
- W3186346120 created "2021-08-02" @default.
- W3186346120 creator A5001081386 @default.
- W3186346120 creator A5006281710 @default.
- W3186346120 creator A5023946565 @default.
- W3186346120 creator A5065499122 @default.
- W3186346120 creator A5076774917 @default.
- W3186346120 date "2021-07-27" @default.
- W3186346120 modified "2023-10-14" @default.
- W3186346120 title "N6-methyladenosine methyltransferases: functions, regulation, and clinical potential" @default.
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