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- W3187875403 endingPage "223" @default.
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- W3187875403 abstract "DNA methylation is an epigenetic modification that contributes to essential biological processes such as retrotransposon silencing, cell differentiation, genomic imprinting and X-chromosome inactivation. DNA methylation generates a stable epigenetic mark associated with silencing of gene expression. Aberrant DNA methylation is associated with the development of different tumor types. Reversing DNA methylation is a rational strategy to restore gene re-expression and induce cell differentiation in cancer. DNA hypomethylating agents is a class of drugs that demonstrated efficacy in different tumors. In this chapter, the classification of DNA hypomethylating agents, their pharmacodynamics and their potential drawbacks will be discussed." @default.
- W3187875403 created "2021-08-16" @default.
- W3187875403 creator A5047899936 @default.
- W3187875403 creator A5067154597 @default.
- W3187875403 date "2021-01-01" @default.
- W3187875403 modified "2023-10-14" @default.
- W3187875403 title "DNA methylation inhibitors: Retrospective and perspective view" @default.
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