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- W3188643573 abstract "Tucatinib (TUC), a highly selective HER2-directed TKI with minimal EGFR inhibition approved for HER2+ metastatic breast cancer, is being developed for patients (pts) with metastatic colorectal cancer (mCRC) and other GI tumors. In GEC xenograft models, dual targeting of HER2 with TUC and trastuzumab (Tras) showed superior activity to either agent alone. Interim results from the MOUNTAINEER study have shown promising activity for TUC and Tras in HER2+ mCRC." @default.
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- W3188643573 date "2021-09-01" @default.
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- W3188643573 title "1434TiP MOUNTAINEER-02: Phase II/III study of tucatinib, trastuzumab, ramucirumab, and paclitaxel in previously treated HER2+ gastric or gastroesophageal junction adenocarcinoma (GEC): Trial in progress" @default.
- W3188643573 doi "https://doi.org/10.1016/j.annonc.2021.08.1543" @default.
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