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- W3197443880 endingPage "213" @default.
- W3197443880 startingPage "175" @default.
- W3197443880 abstract "Since the discovery of the proto-oncogene Wnt1 (Int1) in 1982, WNT signaling has been identified as one of the most important pathways that regulates a wide range of fundamental developmental and physiological processes in multicellular organisms. The canonical WNT signaling pathway depends on the stabilization and translocation of β-catenin and plays important roles in development and homeostasis. The WNT/planar cell polarity (WNT/PCP) signaling, also known as one of the β-catenin-independent WNT pathways, conveys directional information to coordinate polarized cell behaviors. Similar to WNT/β-catenin signaling, disruption or aberrant activation of WNT/PCP signaling also underlies a variety of developmental defects and cancers. However, the pharmacological targeting of WNT/PCP signaling for therapeutic purposes remains largely unexplored. In this review, we briefly discuss WNT/PCP signaling in development and disease and summarize the known drugs/inhibitors targeting this pathway." @default.
- W3197443880 created "2021-09-13" @default.
- W3197443880 creator A5018244700 @default.
- W3197443880 creator A5033378934 @default.
- W3197443880 creator A5070463001 @default.
- W3197443880 date "2021-01-01" @default.
- W3197443880 modified "2023-10-01" @default.
- W3197443880 title "An Overview of Potential Therapeutic Agents Targeting WNT/PCP Signaling" @default.
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