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- W3200803057 endingPage "113856" @default.
- W3200803057 startingPage "113856" @default.
- W3200803057 abstract "Retinol-binding protein 4 (RBP4) is a serum protein that transports Vitamin A. RBP4 is correlated with numerous diseases and metabolic syndromes, including insulin resistance in type 2 diabetes, cardiovascular diseases, obesity, and macular degeneration. Recently, RBP4 antagonists and protein synthesis inhibitors are under development to regulate the effect of RBP4. Several RBP4 antagonists, especially BPN-14136, have demonstrated promising safety profiles and potential therapeutic benefits in animal studies. Two RBP4 antagonists, specifically tinlarebant (Belite Bio) and STG-001 (Stargazer) are currently undergoing clinical trials. Some antidiabetic drugs and nutraceuticals have been reported to reduce RBP4 expression, but more clinical data is needed to evaluate their therapeutical benefits. As regulating RBP4 levels or its activities would benefit a wide range of patients, further research is highly recommended to develop clinically useful RBP4 antagonists or protein synthesis inhibitors." @default.
- W3200803057 created "2021-09-27" @default.
- W3200803057 creator A5035669509 @default.
- W3200803057 creator A5083717295 @default.
- W3200803057 date "2021-12-01" @default.
- W3200803057 modified "2023-10-16" @default.
- W3200803057 title "Retinol binding protein 4 antagonists and protein synthesis inhibitors: Potential for therapeutic development" @default.
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- W3200803057 doi "https://doi.org/10.1016/j.ejmech.2021.113856" @default.
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