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- W3201110329 abstract "Abstract Ebselen is a well-known synthetic compound mimicking glutathione peroxidase (GPx), which catalyses some vital reactions that protect against oxidative damage. Based on a large number of in vivo and in vitro studies, various mechanisms have been proposed to explain its actions on multiple targets. It targets thiol-related compounds, including cysteine, glutathione, and thiol proteins (e.g., thioredoxin and thioredoxin reductase). Owing to this, ebselen is a unique multifunctional agent with important effects on inflammation, apoptosis, oxidative stress, cell differentiation, immune regulation and neurodegenerative disease, with anti-microbial, detoxifying and anti-tumour activity. This review summarises the current understanding of the multiple biological processes and molecules targeted by ebselen, and its pharmacological applications." @default.
- W3201110329 created "2021-09-27" @default.
- W3201110329 creator A5001288058 @default.
- W3201110329 creator A5026086160 @default.
- W3201110329 creator A5026178999 @default.
- W3201110329 creator A5031800532 @default.
- W3201110329 creator A5042241049 @default.
- W3201110329 creator A5053196992 @default.
- W3201110329 creator A5058485605 @default.
- W3201110329 creator A5072162314 @default.
- W3201110329 date "2021-01-01" @default.
- W3201110329 modified "2023-09-28" @default.
- W3201110329 title "Ebselen, a multi-target compound: its effects on biological processes and diseases" @default.
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