Matches in SemOpenAlex for { <https://semopenalex.org/work/W3203457175> ?p ?o ?g. }
- W3203457175 endingPage "14010" @default.
- W3203457175 startingPage "13980" @default.
- W3203457175 abstract "We review progress in the application of fragment-based drug discovery (FBDD) to epigenetic drug discovery (EPIDD) targeted at epigenetic writer and eraser enzymes as well as reader domains over the last 15 years. The greatest successes to date are in prospecting for bromodomain binding ligands. From a diverse array of fragment hits, multiple potent and selective compounds ensued, including the oncology clinical candidates mivebresib, ABBV-744, pelabresib, and PLX51107." @default.
- W3203457175 created "2021-10-11" @default.
- W3203457175 creator A5030865226 @default.
- W3203457175 creator A5049101460 @default.
- W3203457175 creator A5064355287 @default.
- W3203457175 date "2021-09-30" @default.
- W3203457175 modified "2023-10-16" @default.
- W3203457175 title "From Hit Seeking to Magic Bullets: The Successful Union of Epigenetic and Fragment Based Drug Discovery (EPIDD + FBDD)" @default.
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