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- W3208174929 abstract "Proteolysis-Targeting Chimera Technology In article number 2102555, Hong-yu Li, Haojie Huang, and co-workers demonstrate a new approach, oligonucleotide-based proteolysis-targeting chimera (O'PROTAC), to degrade “undruggable” transcriptional factors (TFs) via the ubiquitin-proteasome system. O'PROTAC is designed by employing the TF-uniquely-recognized DNA sequence as natural “ligand”. The programmability of O'PROTAC makes it an attractive arsenal to target TFs for treatment of diseases including cancer." @default.
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- W3208174929 date "2021-10-01" @default.
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- W3208174929 title "Destruction of DNA‐Binding Proteins by Programmable Oligonucleotide PROTAC (O'PROTAC): Effective Targeting of LEF1 and ERG (Adv. Sci. 20/2021)" @default.
- W3208174929 doi "https://doi.org/10.1002/advs.202170136" @default.
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