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- W3210731903 abstract "Nowadays, nitrogenous heterocyclic molecules have attracted a great deal of interest among medicinal chemists. Among these potential heterocyclic drugs, benzimidazole scaffolds are considerably prevalent. Due to their isostructural pharmacophore of naturally occurring active biomolecules, benzimidazole derivatives have significant importance as chemotherapeutic agents in diverse clinical conditions. Researchers have synthesized plenty of benzimidazole derivatives in the last decades, amidst a large share of these compounds exerted excellent bioactivity against many ailments with outstanding bioavailability, safety, and stability profiles. In this comprehensive review, we have summarized the bioactivity of the benzimidazole derivatives reported in recent literature (2012-2021) with their available structure-activity relationship. Compounds bearing benzimidazole nucleus possess broad-spectrum pharmacological properties ranging from common antibacterial effects to the world's most virulent diseases. Several promising therapeutic candidates are undergoing human trials, and some of these are going to be approved for clinical use. However, notable challenges, such as drug resistance, costly and tedious synthetic methods, little structural information of receptors, lack of advanced software, and so on, are still viable to be overcome for further research." @default.
- W3210731903 created "2021-11-08" @default.
- W3210731903 creator A5009375949 @default.
- W3210731903 creator A5020229643 @default.
- W3210731903 creator A5031165279 @default.
- W3210731903 creator A5031472760 @default.
- W3210731903 creator A5076056592 @default.
- W3210731903 creator A5083168839 @default.
- W3210731903 date "2021-11-03" @default.
- W3210731903 modified "2023-10-05" @default.
- W3210731903 title "A Comprehensive Account on Recent Progress in Pharmacological Activities of Benzimidazole Derivatives" @default.
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