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- W32386813 abstract "Current systemic therapies for breast cancer are often limited by their non-specific mechanism of action, unwanted toxicities on normal tissues and short-term efficacy due to the emergence of drug resistance. Identification of the molecular alterations in key proteins involved in breast cancer cell proliferation and survival resulted in development of various signal transduction inhibitors as new treatment strategy. Preclinical data support the use of these agents in breast cancer, including estrogen receptor positive breast cancer patients in which signalling inhibitors might prevent or treat resistance to endocrine therapy. These compounds have generally shown an acceptable toxicity profile. However, little clinical activity of signalling inhibitors as monotherapy in breast cancer patients has been reported up to now. Furthermore, the preliminary results of clinical trials of combinations of signalling inhibitors and endocrine therapies published to day are rather disappointing. These negative findings are likely due to the occurrence of mechanisms of resistance to these drugs." @default.
- W32386813 created "2016-06-24" @default.
- W32386813 creator A5003014678 @default.
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- W32386813 creator A5054637398 @default.
- W32386813 creator A5081955195 @default.
- W32386813 creator A5089331461 @default.
- W32386813 date "2009-01-01" @default.
- W32386813 modified "2023-10-18" @default.
- W32386813 title "Signal Transduction Inhibitors in the Treatment of Breast Cancer" @default.
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