Matches in SemOpenAlex for { <https://semopenalex.org/work/W40325719> ?p ?o ?g. }
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- W40325719 abstract "γ-Aminobutyric acid type A receptors (GABAARs) are the principal mediators of fast synaptic inhibition in the brain as well as the low persistent extrasynaptic inhibition, both of which are fundamental to proper brain function. Thus unsurprisingly, deficits in GABAARs are implicated in a number of neurological disorders and diseases. The complexity of GABAAR regulation is determined not only by the heterogeneity of these receptors but also by its posttranslational modifications, the foremost, and best characterized of which is phosphorylation. This review will explore the details of this dynamic process, our understanding of which has barely scratched the surface. GABAARs are regulated by a number of kinases and phosphatases, and its phosphorylation plays an important role in governing its trafficking, expression, and interaction partners. Here, we summarize the progress in understanding the role phosphorylation plays in the regulation of GABAARs. This includes how phosphorylation can affect the allosteric modulation of GABAARs, as well as signaling pathways that affect GABAAR phosphorylation. Finally, we discuss the dysregulation of GABAAR phosphorylation and its implication in disease processes." @default.
- W40325719 created "2016-06-24" @default.
- W40325719 creator A5006927586 @default.
- W40325719 creator A5020338130 @default.
- W40325719 creator A5037112586 @default.
- W40325719 creator A5039050340 @default.
- W40325719 date "2015-01-01" @default.
- W40325719 modified "2023-10-05" @default.
- W40325719 title "Regulation of GABAARs by Phosphorylation" @default.
- W40325719 cites W1499733802 @default.
- W40325719 cites W1515260227 @default.
- W40325719 cites W1516599165 @default.
- W40325719 cites W1524203275 @default.
- W40325719 cites W1551663317 @default.
- W40325719 cites W1555899391 @default.
- W40325719 cites W1556008197 @default.
- W40325719 cites W1557205789 @default.
- W40325719 cites W1559776259 @default.
- W40325719 cites W1563745248 @default.
- W40325719 cites W1569931447 @default.
- W40325719 cites W1594117694 @default.
- W40325719 cites W1597102052 @default.
- W40325719 cites W1607645391 @default.
- W40325719 cites W1627446849 @default.
- W40325719 cites W1661938295 @default.
- W40325719 cites W1672480124 @default.
- W40325719 cites W1691674240 @default.
- W40325719 cites W1701778517 @default.
- W40325719 cites W1705218924 @default.
- W40325719 cites W1718935338 @default.
- W40325719 cites W1781472042 @default.
- W40325719 cites W1783438623 @default.
- W40325719 cites W1815276265 @default.
- W40325719 cites W1845046061 @default.
- W40325719 cites W1892249233 @default.
- W40325719 cites W1951170463 @default.
- W40325719 cites W1957331510 @default.
- W40325719 cites W1964347457 @default.
- W40325719 cites W1965081959 @default.
- W40325719 cites W1966087347 @default.
- W40325719 cites W1966331279 @default.
- W40325719 cites W1966968864 @default.
- W40325719 cites W1967075253 @default.
- W40325719 cites W1967516237 @default.
- W40325719 cites W1968700646 @default.
- W40325719 cites W1969088566 @default.
- W40325719 cites W1969520694 @default.
- W40325719 cites W1970851102 @default.
- W40325719 cites W1973115552 @default.
- W40325719 cites W1976495250 @default.
- W40325719 cites W1976763493 @default.
- W40325719 cites W1977892054 @default.
- W40325719 cites W1978022925 @default.
- W40325719 cites W1985946118 @default.
- W40325719 cites W1988394046 @default.
- W40325719 cites W1988749472 @default.
- W40325719 cites W1989916543 @default.
- W40325719 cites W1989979738 @default.
- W40325719 cites W1991714532 @default.
- W40325719 cites W1992291881 @default.
- W40325719 cites W1993480664 @default.
- W40325719 cites W1993874939 @default.
- W40325719 cites W1993901712 @default.
- W40325719 cites W1994261508 @default.
- W40325719 cites W1994264681 @default.
- W40325719 cites W1995842626 @default.
- W40325719 cites W1996927830 @default.
- W40325719 cites W1997425969 @default.
- W40325719 cites W1998050348 @default.
- W40325719 cites W1999383552 @default.
- W40325719 cites W1999704138 @default.
- W40325719 cites W2000079550 @default.
- W40325719 cites W2000087227 @default.
- W40325719 cites W2000757833 @default.
- W40325719 cites W2000917831 @default.
- W40325719 cites W2001162506 @default.
- W40325719 cites W2003408651 @default.
- W40325719 cites W2004998882 @default.
- W40325719 cites W2009063652 @default.
- W40325719 cites W2009782005 @default.
- W40325719 cites W2010890416 @default.
- W40325719 cites W2011469680 @default.
- W40325719 cites W2012785062 @default.
- W40325719 cites W2013775967 @default.
- W40325719 cites W2013903929 @default.
- W40325719 cites W2014038449 @default.
- W40325719 cites W2014271878 @default.
- W40325719 cites W2015227366 @default.
- W40325719 cites W2016321438 @default.
- W40325719 cites W2017027505 @default.
- W40325719 cites W2017807856 @default.
- W40325719 cites W2018547231 @default.
- W40325719 cites W2021677873 @default.
- W40325719 cites W2022802363 @default.
- W40325719 cites W2023863818 @default.
- W40325719 cites W2024801162 @default.
- W40325719 cites W2025670735 @default.
- W40325719 cites W2025672307 @default.