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- W4200399276 abstract "Poly(ADP-ribose) polymerase (PARP) inhibitors (PARPi) are now a first-line maintenance treatment in ovarian cancer and have been approved in other cancer types, including breast, pancreatic and prostate. Despite their efficacy, and as is the case for other targeted therapies, resistance to PARPi has been reported clinically and is generating a growing patient population of unmet clinical need. Here, we discuss the mechanisms of resistance that have been described in pre-clinical models and focus on those that have been already identified in the clinic, highlighting the key challenges to fully characterise the clinical landscape of PARPi resistance and proposing ways of preventing and overcoming it." @default.
- W4200399276 created "2021-12-31" @default.
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- W4200399276 creator A5083333226 @default.
- W4200399276 date "2021-12-23" @default.
- W4200399276 modified "2023-10-14" @default.
- W4200399276 title "Preventing and Overcoming Resistance to PARP Inhibitors: A Focus on the Clinical Landscape" @default.
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