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- W4205122795 endingPage "319" @default.
- W4205122795 startingPage "319" @default.
- W4205122795 abstract "Human protozoan diseases represent a serious health problem worldwide, affecting mainly people in social and economic vulnerability. These diseases have attracted little investment in drug discovery, which is reflected in the limited available therapeutic arsenal. Authorized drugs present problems such as low efficacy in some stages of the disease or toxicity, which result in undesirable side effects and treatment abandonment. Moreover, the emergence of drug-resistant parasite strains makes necessary an even greater effort to develop safe and effective antiparasitic agents. Among the chemotypes investigated for parasitic diseases, the indole nucleus has emerged as a privileged molecular scaffold for the generation of new drug candidates. In this review, the authors provide an overview of the indole-based compounds developed against important parasitic diseases, namely malaria, trypanosomiasis and leishmaniasis, by focusing on the design, optimization and synthesis of the most relevant synthetic indole scaffolds recently reported." @default.
- W4205122795 created "2022-01-25" @default.
- W4205122795 creator A5063797318 @default.
- W4205122795 creator A5087842000 @default.
- W4205122795 date "2022-01-05" @default.
- W4205122795 modified "2023-10-14" @default.
- W4205122795 title "Recent Progress in the Development of Indole-Based Compounds Active against Malaria, Trypanosomiasis and Leishmaniasis" @default.
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