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- W4206024975 abstract "Polymersomes (Ps) are defined as artificial vesicles, resulting from the assembly of synthetic amphiphilic copolymer blocks, capable of carrying and releasing drugs. Compared to other vesicular nanovectors, such as liposomes or nanoparticles, they are very versatile because of the possibility to encapsulate drugs of different nature, such as hydrophilic, lipophilic, DNA and RNA molecules, and vaccines. It is also possible to functionalize their surface, by increasing their transport across biological membranes and optimizing the pharmacokinetics and biodistribution of drugs conjugated to them at target site. Also, Ps possesses remarkable colloidal stability, tunable membrane permeability, excellent robustness, and relatively long blood circulation times attributable to their high biocompatibility with biological systems. In recent years, these nanovectors have received significant research interest because they could mediate drug release in response to a series of internal biological stimuli (pH, redox potential, and glucose concentration) and external physical stimuli (temperature, light, and ultrasound), which can induce significant changes in the structure of the Ps with consequent destruction of the membrane and drug release. The advantages, offered in terms of therapeutic efficacy and reduction of side effects, make these carriers excellent delivery systems for drugs but also for medical imaging and diagnostics. Therefore, the aim of this chapter is to investigate the strategies, progresses, and advantages of using Ps as carriers for stimuli-responsive drug delivery." @default.
- W4206024975 created "2022-01-25" @default.
- W4206024975 creator A5001037825 @default.
- W4206024975 creator A5030059410 @default.
- W4206024975 creator A5086524999 @default.
- W4206024975 date "2022-01-01" @default.
- W4206024975 modified "2023-09-26" @default.
- W4206024975 title "Polymersomes as a promising vehicle for controlled drug delivery" @default.
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