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- W4210967589 endingPage "139" @default.
- W4210967589 startingPage "127" @default.
- W4210967589 abstract "Bile salts are amphipathic molecules conjugated to glycine or taurine and display detergent properties. They play essential roles in promoting fat digestion and absorption or excretion of cholesterol, lipids, lipophilic nutrients, and other hydrophobic compounds in the liver and the intestine. Enterohepatic circulation of bile salts is mediated by specific transporters, most of which are integral plasma membrane proteins and are expressed in hepatocytes and enterocytes in a polarized manner. This chapter focuses on the mechanisms that regulate the expression of bile salt transporters at the transcriptional level. The dependence of the transcriptional activity of most nuclear and steroid receptors on specific ligands allows them to monitor intracellular environment and to elicit rapid transcriptional responses to changes in the concentrations of specific compounds. Transport and metabolism of exogenous compounds, such as drugs, nutrients, and environmental xenobiotics, bear many similarities to those of endogenous bile salts." @default.
- W4210967589 created "2022-02-13" @default.
- W4210967589 creator A5042283235 @default.
- W4210967589 creator A5080077380 @default.
- W4210967589 creator A5089543992 @default.
- W4210967589 date "2014-08-08" @default.
- W4210967589 modified "2023-10-10" @default.
- W4210967589 title "Bile Salt Transporters" @default.
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