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- W4211036692 abstract "Expressed primarily in cardiac myocytes, the hERG channel (Kv11.1) is a voltage-gated potassium channel that facilitates a repolarizing K+ current during the cardiac action potential (CAP). In response to changes in membrane potential, the hERG channel undergoes transitions from closed to open and inactivated states. Utilizing atomistic molecular modeling and docking simulations, we aim to assess the state-specific binding of drugs to the hERG channel utilizing structural models of open and inactivated hERG channels." @default.
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- W4211036692 date "2022-02-01" @default.
- W4211036692 modified "2023-10-14" @default.
- W4211036692 title "Exploring drug arrythmogenicity via atomistic simulations of state-specific hERG-channel block" @default.
- W4211036692 doi "https://doi.org/10.1016/j.bpj.2021.11.2457" @default.
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