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- W4211064888 endingPage "478" @default.
- W4211064888 startingPage "445" @default.
- W4211064888 abstract "Nuclear molecular imaging is fueled by a diverse set of radiopharmaceuticals that enable the visualization of biological targets and processes in normal and disease states. Over the last 40–50 years, a rich set of radiochemistry reactions has been amassed to prepare a panoply of radiopharmaceuticals. A diverse set of positron-emitting radionuclides provides an array of physical and chemical properties that may be exploited to radiolabel small molecules to nanoparticles. Carbon, nitrogen, oxygen, and fluorine are elements that are commonly found in biomolecules and drug candidates. These four elements have radioisotopes that are near pure positron emitters with suitable imaging properties. Radiometals, typically with longer half-lives, may be conjugated to molecular agents with similar biological half-life. Creative chemistry approaches enable the preparation of radiopharmaceuticals and labeled drugs for in vivo evaluation. Herein, an overview of positron emission tomography radiochemistry is presented, highlighting the significant advances in the field covering diverse chemical and biological space." @default.
- W4211064888 created "2022-02-13" @default.
- W4211064888 creator A5074856469 @default.
- W4211064888 date "2021-01-01" @default.
- W4211064888 modified "2023-09-26" @default.
- W4211064888 title "PET Radiochemistry" @default.
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