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- W4211216385 startingPage "169" @default.
- W4211216385 abstract "In 1987, zidovudine became the first approved agent in the United States for the treatment of human immunodeficiency virus type 1 (HIV-1) infection. Almost 30 years later, more than 26 additional agents in six drug classes have been approved. These include nucleoside/nucleotide reverse transcriptase inhibitors (NRTIs), non-nucleoside reverse transcriptase inhibitors (NNRTIs), protease inhibitors (PIs), a fusion inhibitor (entry inhibitor), a chemokine coreceptor antagonist (entry inhibitor), integrase strand transfer inhibitors (Table 1), and pharmacokinetic enhancers. This success is the result of a prodigious effort to dissect the virus’ replication cycle and the virion's interaction with its CD4 target cells to identify promising drug targets. It also illustrates the interdependency of the drug development process, knowledge of disease pathogenesis, and use of sensitive therapeutic monitoring tools like plasma HIV-1 RNA levels and drug resistance testing." @default.
- W4211216385 created "2022-02-13" @default.
- W4211216385 creator A5018295987 @default.
- W4211216385 creator A5063382165 @default.
- W4211216385 creator A5064182369 @default.
- W4211216385 date "2016-03-07" @default.
- W4211216385 modified "2023-09-26" @default.
- W4211216385 title "Antiretroviral Agent" @default.
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