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- W4220779188 abstract "Highly active antiretroviral therapy currently used for HIV/AIDS has significantly increased the life expectancy of HIV-infected individuals. It has also improved the quality of life, reduced mortality, and decreased the incidence of AIDS and HIV-related conditions. Currently, however, affected individuals are typically on a lifetime course of several therapeutic drugs, all with the potential for associated toxicity and emergence of resistance. This calls for development of novel, potent, and broad anti-HIV agents able to stop the spread of HIV/AIDS. Significant progress has been made toward identification of anti-HIV-1 broadly neutralizing antibodies (bNAbs). However, antibody-based drugs are costly to produce and store. Administration (by injection only) and other obstacles limit clinical use. In recent years, several highly promising small-molecule HIV-1 entry inhibitors targeting the epitopes of bNAbs have been developed. These newly developed compounds are the focus of the present article." @default.
- W4220779188 created "2022-04-03" @default.
- W4220779188 creator A5004434095 @default.
- W4220779188 creator A5064289593 @default.
- W4220779188 creator A5069302796 @default.
- W4220779188 date "2022-05-01" @default.
- W4220779188 modified "2023-09-23" @default.
- W4220779188 title "Small-molecule HIV-1 entry inhibitors targeting the epitopes of broadly neutralizing antibodies" @default.
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