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- W4224290038 abstract "The development of new and effective therapeutics is reliant on the ability to study the underlying mechanisms of potential drug targets in live cells and multicellular systems. A persistent challenge in many drug development programmes is poor selectivity, which can obscure the mechanisms involved and lead to poorly understood modes of action. In efforts to improve our understanding of these complex processes, small molecule inhibitors have been developed in which their OFF/ON therapeutic activity can be toggled using light. Photopharmacology is devoted to using light to modulate drugs. Herein, we highlight the recent progress made towards the development of light-responsive small molecule inhibitors of selected enzymatic targets. Given the size of this field, literature from 2015 onwards has been reviewed." @default.
- W4224290038 created "2022-04-26" @default.
- W4224290038 creator A5000996540 @default.
- W4224290038 creator A5015128267 @default.
- W4224290038 creator A5035703153 @default.
- W4224290038 date "2022-04-21" @default.
- W4224290038 modified "2023-10-01" @default.
- W4224290038 title "Photoresponsive Small Molecule Inhibitors for the Remote Control of Enzyme Activity" @default.
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