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- W4237598678 abstract "Significant improvement in metabolic stability on the pyrazolopiperidine scaffold over the original series were achieved and this stability improvement translated in an improved in vivo efficacy." @default.
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- W4237598678 date "2010-06-01" @default.
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- W4237598678 title "Discovery of a novel sulfonamide-pyrazolopiperidine series as potent and efficacious γ-secretase inhibitors (Part II)" @default.
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- W4237598678 doi "https://doi.org/10.1016/j.bmcl.2010.04.148" @default.
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