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- W4238059486 abstract "The optimization of low-potency leads into drugs is often accompanied by an increase in molecular weight (Mr) and lipophilicity, as a consequence of affinity enhancement. Hits with affinity at μM levels discovered by screening leadlike libraries allow scope for this optimization process, as shown schematically by the distributions of Mr for a leadlike library (1), oral drugs (2), and a typical combinatorial chemistry library (3). y=percentage with a particular molecular weight." @default.
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- W4238059486 date "1999-12-16" @default.
- W4238059486 modified "2023-09-28" @default.
- W4238059486 title "The Design of Leadlike Combinatorial Libraries" @default.
- W4238059486 doi "https://doi.org/10.1002/(sici)1521-3773(19991216)38:24<3743::aid-anie3743>3.3.co;2-l" @default.
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