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- W4241624521 abstract "This review deals with a newly-developed category of antithrombotic drugs – the direct thrombin inhibitors. These agents interact with thrombin and block its catalytic activity on fibrinogen, platelets and other substrates. Heparin and its derivatives (low molecular weight heparins and the active pentasaccharide) inhibit thrombin and/or other coagulation serine proteases indirectly via antithrombin, and the warfarin-type drugs interfere with the synthesis of the precursors of the coagulation serine proteases. The direct thrombin inhibitors approved for clinical use at present (lepirudin, desirudin, bivalirudin, argatroban) and another in the advanced clinical testing stage (melagatran/ximelagatran), are the subject of this review. The chemical structure; kinetics of thrombin inhibition; pharmacokinetics and clinical use of each of these is discussed." @default.
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- W4241624521 date "2003-01-01" @default.
- W4241624521 modified "2023-09-24" @default.
- W4241624521 title "Direct thrombin inhibitors" @default.
- W4241624521 doi "https://doi.org/10.1517/eoph.4.5.653.22217" @default.
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