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- W4242107009 endingPage "124" @default.
- W4242107009 startingPage "106" @default.
- W4242107009 abstract "This chapter presents an overview of opioid analgesics and narcotic antagonists. Oral administration is the method most often used with opioid analgesics because it is noninvasive, convenient and easy to titrate. In chronic pain, oral opioid formulations that provide longer durations of effect are preferred, because they provide more stable pain control, better tolerability, and increased convenience, patient options, and flexibility. Dextromethorphan is a noncompetitive antagonist at N-methyl-D-aspartate (NMDA) receptors. It is antitussive and has antihyperalgesic effects. In 25 volunteers, intravenous dextromethorphan 0.5 mg/kg significantly reduced areas of established hyperalgesia after tissue injury by 39% and prevented the development of further hyperalgesia. There was large inter-subject variability in the timing of this effect, with an average duration of 2 hours in relation to peak serum concentration. In this chapter, routes of administration of opioids are explained in detail. Opioid receptor agonists are discussed. An overview of levo-α-acetylmethadol (LAAM), methadone, buprenorphine, nalbuphine, and nalmefene is also presented in the chapter." @default.
- W4242107009 created "2022-05-12" @default.
- W4242107009 creator A5059131102 @default.
- W4242107009 creator A5087957539 @default.
- W4242107009 date "2008-01-01" @default.
- W4242107009 modified "2023-10-16" @default.
- W4242107009 title "Opioid analgesics and narcotic antagonists" @default.
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