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- W4246706954 abstract "We have discovered new chemical compounds that are characterized as Kir channel inhibitors of the Aedes aegypti mosquito. This is important as the Ae. aegypti mosquito is the primary vector for Zika virus (ZIKV), Dengue virus (DENV) and chikungunya virus (CHIKV). Traditional mosquitocides are plagued with significant resistance and developing new compounds with novel mechanisms of action are vitally important. Lastly, we show that our compounds are potent larvicides against pyrethroid-susceptible and pyrethroid-resistant strains." @default.
- W4246706954 created "2022-05-12" @default.
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- W4246706954 date "2020-07-20" @default.
- W4246706954 modified "2023-10-17" @default.
- W4246706954 title "Further SAR on the (Phenylsulfonyl)piperazine Scaffold as Inhibitors of the Aedes Aegypti Kir1 (AeKir) Channel and Larvicides" @default.
- W4246706954 doi "https://doi.org/10.26434/chemrxiv.12662690" @default.
- W4246706954 hasPublicationYear "2020" @default.
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