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- W4255656421 abstract "<div>Conjugation of the transitionstate-cation analogue DANA to polymeric scaffolds led to highly potent inhibitors of bacterial sialidases. Each clustered DANA on the polymers saw its inhibitory potency for S. pneumoniae or B. thetaiotaomicron sialidases improved by more than four orders of magnitude. This extends the multivalent concept to this important class of enzymes.</div><div><br></div>" @default.
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- W4255656421 date "2020-09-29" @default.
- W4255656421 modified "2023-10-17" @default.
- W4255656421 title "Polymers of a Transition-State Sialyl Cation Strongly Inhibit Bacterial Sialidases." @default.
- W4255656421 doi "https://doi.org/10.26434/chemrxiv.13013291.v1" @default.
- W4255656421 hasPublicationYear "2020" @default.
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