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- W4256503820 abstract "Two neurokinin B (NKB) analogs, [Gly6]-NKB [3–10] and [Arg3, d-Ala6]-NKB [3–10], were tested for agonistic activity as well as for their ability to antagonize the myotropic actions of NKB, neurokinin A, substance P, physalaemin and eledoisin in isolated guinea-pig ileum, guinea-pig urinary bladder, rat duodenum, rat vas deferens and rat portal vein. [Gly6]-NKB [3–10] in the guinea-pig ileum and rat portal vein and [Arg3, d-Ala6]-NKB [3–10] in the guinea-pig ileum were found to be the first specific and competitive antagonists against NKB." @default.
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- W4256503820 date "1987-01-01" @default.
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- W4256503820 title "Tachykinin Antagonist I: Specific, Competitive and Tissue-Selective Neurokinin B Antagonists on Contractile Activity in Smooth Muscles" @default.
- W4256503820 doi "https://doi.org/10.1016/s0021-5198(19)43380-5" @default.
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