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- W4282972239 endingPage "2224" @default.
- W4282972239 startingPage "2209" @default.
- W4282972239 abstract "Abstract: P2Y receptors (P2YRs) are G protein-coupled receptors that are activated by extracellular nucleotides. The P2Y6 receptor (P2Y6R) is specifically activated by UDP, causing PKC activation and intracellular calcium ion release through the PLC pathway. Based on receptor tissue distribution and related pathways, several studies have reported that P2Y6R plays a physiological role in mediating inflammation, which suggests that P2Y6R could be a promising molecular target for the treatment of inflammatory diseases. In the past ten years, several P2Y6R antagonists have been discovered as new therapeutic strategies for inflammatory diseases. In this article, we systematically summarize the role of P2Y6R in inflammation and highlight the anti-inflammatory mechanism of a key P2Y6R antagonist, MRS2578. Insight into recent progress on the discovery of P2Y6R antagonists is also discussed." @default.
- W4282972239 created "2022-06-17" @default.
- W4282972239 creator A5013382930 @default.
- W4282972239 creator A5026559726 @default.
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- W4282972239 creator A5051198814 @default.
- W4282972239 creator A5062094478 @default.
- W4282972239 creator A5091614841 @default.
- W4282972239 date "2023-05-01" @default.
- W4282972239 modified "2023-10-15" @default.
- W4282972239 title "P2Y6R: A Promising New Target in Inflammatory Diseases and Advances in its Antagonists" @default.
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