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- W4285358733 abstract "Novos alvos terapêuticos para artrite reumatoide (AR) e outras doenças reumáticas imunomediadas (DRIM) vêm sendo elucidados, entre eles a Janus quinases (JAKs). Essas estruturas são essenciais para a sinalização intracelular (via JAK-STAT) em resposta as muitas citocinas envolvidas na imunopatogênese das DRIM. Os inibidores de JAK (iJAK) têm se consolidado como um tratamento altamente eficaz, ganhando cada vez mais espaço no arsenal terapêutico da AR. O presente artigo tem como objetivo apresentar uma atualização dos principais aspectos relacionados ao mecanismo de ação, eficácia e segurança do iJAKs, com ênfase no tratamento de pacientes com AR. Unitermos: Artropatias inflamatórias. Artrite reumatoide. Doenças reumáticas imunomediadas. Inibidores de JAK. Janus quinases. JAK-STAT. Drogas modificadoras do curso da doença sintéticas alvo específicas." @default.
- W4285358733 created "2022-07-14" @default.
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- W4285358733 date "2021-09-30" @default.
- W4285358733 modified "2023-10-18" @default.
- W4285358733 title "Inibidores de Janus quinases (iJAK)" @default.
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- W4285358733 doi "https://doi.org/10.46833/reumatologiasp.2021.20.3.40-49" @default.
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