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- W4296011010 abstract "Mitogen-activated protein kinase (MAPK) pathway inhibition activates Unc-51–like autophagy activated kinase (ULK) 1/2 and initiates autophagy to promote survival of RAS/RAF mutant cancers. DCC-3116, a first-in-class potent and selective ULK inhibitor, demonstrated preclinical antitumour activity in combination with MAPK pathway inhibitors. Here, we describe initial DCC-3116 monotherapy results from an ongoing phase I study." @default.
- W4296011010 created "2022-09-17" @default.
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- W4296011010 date "2022-09-01" @default.
- W4296011010 modified "2023-09-28" @default.
- W4296011010 title "450O Initial monotherapy results of a phase I first-in-human study of ULK1/2 inhibitor DCC-3116 alone and in combination with MAPK pathway inhibition" @default.
- W4296011010 doi "https://doi.org/10.1016/j.annonc.2022.07.579" @default.
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